Cerivastatin
Cerivastatin tablets
What are cerivastatin tablets?
CERIVASTATIN (Baycol™) blocks the body's ability to make cholesterol. Cerivastatin can help lower blood cholesterol for patients who are at risk of getting heart disease or a stroke. It is only for patients whose cholesterol level is not controlled by diet. It is not a cure.
NOTE: This drug is discontinued in the United States.
What should my health care professional know before I take cerivastatin?
They need to know if you have any of these conditions:
an alcohol problem
any hormone disorder (such as diabetes, under-active thyroid)
blood salt imbalance
infection
kidney disease
liver disease
low blood pressure
muscle disorder or condition
recent surgery
seizures (convulsions)
severe injury
an unusual or allergic reaction to cerivastatin, other medicines, foods, dyes, or preservatives
pregnant or trying to get pregnant
breast-feeding
How should I take this medicine?
Take cerivastatin tablets by mouth. Follow the directions on the prescription label. Swallow the cerivastatin with a drink of water. Cerivastatin should be taken at in the evening with or without food. Take your doses at regular intervals. Do not take your medicine more often than directed.
Contact your pediatrician or health care professional regarding the use of this medicine in children. Special care may be needed.
What if I miss a dose?
If you miss a dose, take it as soon as you can. If it is almost time for your next dose, take only that dose. Do not take double or extra doses.
What drug(s) may interact with cerivastatin?
alchohol-containing beverages
amiodarone
bosentan
certain antibiotics such as clarithromycin and erythromycin
cimetidine
diltiazem
grapefruit juice
medicines for fungal infections (examples: fluconazole, itraconazole, ketoconazole, miconazole, voriconazole)
herbal medicines such as red yeast rice
medicines for treating HIV infections
medicines that suppress your immune response (cyclosporine)
medicines to lower cholesterol or triglycerides (examples: cholestyramine, clofibrate, colestipol, fenofibrate, gemfibrozil, niacin)
medicine used to stop early pregnancy (mifepristone, RU-486 or Mifeprex™)
montelukast
nefazodone
niacin
phenytoin
spironolactone
verapamil
Tell your prescriber or health care professional about all other medicines you are taking, including non-prescription medicines, nutritional supplements, or herbal products. Also tell your prescriber or health care professional if you are a frequent user of drinks with caffeine or alcohol, if you smoke, or if you use illegal drugs. These may affect the way your medicine works. Check with your health care professional before stopping or starting any of your medicines.
What should I watch for while taking cerivastatin?
Visit your prescriber or health care professional for regular checks on your progress. You will need to have regular tests to make sure your liver is working properly.
Tell your prescriber or health care professional as soon as you can if you get any unexplained muscle pain, tenderness, or weakness, especially if you also have a fever and tiredness.
Cerivastatin is only part of a total cholesterol-lowering program. Your physician or dietician can suggest a low-cholesterol and low-fat diet that will reduce your risk of getting heart and blood vessel disease. Avoid alcohol and smoking, and keep a proper exercise schedule.
If you are going to have surgery tell your prescriber or health care professional that you are taking cerivastatin.
What side effects may I notice from taking cerivastatin?
Side effects that you should report to your prescriber or health care professional as soon as possible:
Rare or uncommon:
dark yellow or brown urine
decreased urination, difficulty passing urine
fever
muscle pain, tenderness, cramps, or weakness
redness, blistering, peeling or loosening of the skin, including inside the mouth
skin rash, itching
unusual tiredness or weakness
yellowing of the skin or eyes
Side effects that usually do not require medical attention (report to your prescriber or health care professional if they continue or are bothersome):
diarrhea
difficulty sleepine
gas
headache
joint pain
nausea, vomiting
stomach upset or pain
tiredness
Where can I keep my medicine?
Keep out of the reach of children in a container that small children cannot open.
Store at controlled room temperature between 20 to 25 degrees C (68 to 77 degrees F). Keep container tightly closed. Throw away any unused medicine after the expiration date.
Updated:  
March 21, 2017
Sources:  
U.S. FDA-approved Package Insert